Tag-lite® compound profiling

Cisbio offers a comprehensive compound profiling service covering a wide range of GPCR assays.

Classification of compounds according to their binding affinities is an essential step in the drug discovery process. As a leader in GPCR ligand binding technologies, we will evaluate the binding affinity of your compounds for a receptor of interest, or characterize their mode of action.

Select and send your compounds

Supply from 1 to 50 compounds, such as DMSO stocks solutions. Send your compounds to your local Cisbio testing laboratory.

Select your receptors

You may select any number of receptors from the list below.

Receive your results

A detailed report, including a summary of the testing and a graphical representation, is delivered at the end of the project. A table is provided summarizing the IC50 values for all compounds. With over 20 years of experience in GPCR technologies, our team is committed to delivering quality results in a timely manner.

Receptor family Receptor
Adenosin A2A
Adrenergic Beta 1
Beta 2
Anaphylotoxin C5L2
Angiotensin AT2
Bombesin BB1
BB2
Bradykinin B1
B2
Chemokine CCR5
CXCR4
Cholecystokinin CCK1
CCK2
Class A Orphans GPR1
Dopamine D 1
D 2
D3a
Endothelin ETA
ETB
Ghrelin GHSR1 A
Glucagon GIPR
GLP1
Receptor family Receptor
Histamine H1
H3
Melanocortin MC4
MC5
Cholecystokinin M1
M2
M4
M5
Opioid Delta
Kappa
Orexin OX1
OX2
Parathyroid PTH1
Serotonin 5HT1A
5HT1B
5HT4
Somatostatin SST4
Tackykinin NK1
Vasopressin/Oxytocin V2
RTK EGFR1
Somatostatin SST4
Receptor
Adenosin A2A
Adrenergic Beta 1
Adrenergic Beta 2
Anaphylotoxin C5L2
Angiotensin AT2
Bombesin BB1
Bombesin BB2
Bradykinin B1
Bradykinin B2
Chemokine CCR5
Chemokine CXCR4
Cholecystokinin CCK1
Cholecystokinin CCK2
Class A Orphans GPR1
Dopamine D 1
Dopamine D 2
Dopamine D3a
Endothelin ETA
Endothelin ETB
Ghrelin GHSR1 A
Glucagon GIPR
Glucagon GLP1
Histamine H1
Histamine H3
Melanocortin MC4
Melanocortin MC5
Cholecystokinin M1
Cholecystokinin M2
Cholecystokinin M4
Cholecystokinin M5
Opioid Delta
Opioid Kappa
Orexin OX1
Orexin OX2
Parathyroid PTH1
Serotonin 5HT1A
Serotonin 5HT1B
Serotonin 5HT4
Somatostatin SST4
Tackykinin NK1
Vasopressin/Oxytocin V2
RTK EGFR1
Somatostatin SST4